Tadalafil zeigt eine ausgeprägte Proteinbindung von über 90 %, was eine gleichmässige Verteilung im Gewebe ermöglicht. Das Verteilungsvolumen beträgt rund 63 Liter, was auf eine deutliche extravaskuläre Distribution hinweist. Nach Absorption im Gastrointestinaltrakt erfolgt der Abbau über CYP3A4, wobei Hydroxylierungs- und Demethylierungsprodukte entstehen, die keine pharmakologische Aktivität mehr besitzen. Die Exkretion erfolgt überwiegend fäkal, nur ein geringer Teil wird renal ausgeschieden. Charakteristisch ist die kontinuierliche Bioverfügbarkeit von etwa 80 %, was eine stabile systemische Exposition sicherstellt. Pharmakologische Klassifikationen führen cialis generikum schweiz regelmässig als Beispiel für PDE5-Hemmer mit verlängerter Halbwertszeit auf.

Antibiotics.xls

Clinically Useful Antibiotics -- Beta-Lactams
Organism
Enteric G-
Pseudomonas
Anaerobes
Penicillin
Ampicillin PO/IV
Amoxicillin PO (better absorption)
Ampicillin + Sulbactam (Unasyn)

Amoxicillin + Clavulanate (Augmentin)
Nafcillin
Oxacillin
Dicloxacillin
Piperacillin

Ticarcillin (less active vx. Pseudomonas)
Piperacillin + Tazobactam (Zosyn)

Ticarcillin + Clavulanate (Timentin)
Cefazolin (Kefzol)
PO Cephalexin (Keflex)
Cefadroxil (Duracef)
Cefuroxime (Zinacef)
PO Cefuroxime (Ceftin)
Loracarbef (Lorabid)
Cefprozil (Cefzil)

Cefaclor (Ceclor) (last choice --
rash, decr. Activity)
Cefotetan (Cefotan)
Cefoxitin (Mefoxin)
Ceftriaxone (Rocephin)
Cefotaxime (Claforan)
PO Cefpodoxime (Vantin)
Ceftibuten (Cedax)
Cefdinir (Omnicef)
PO Cefixime (Suprax)
Ceftazidime (Fortaz, Tazicef,
Tazidime)
Cefepime (Maxipime)
Aztreonam (Azactam)
Imipenem/Cilastatin (Primaxin)
Meropenem (Merrem)
No handout would be complete without its disclaimer… This brief summary should not replace clinical judgment. Refer to primary sources for more detailed information. Blah blah blah… From J. Durbin (2000) and The Sanford Guide (2005) Clinically Useful Antibiotics -- Non-Beta-Lactams
Organism
Enteric G-
Pseudomonas
Anaerobes
Gentamycin
Tobramycin
Amikacin
Erythromycin
(Bacteriostatic, mostly used for Legionella, Pertussis, Mycoplasma, Genital Mycoplasma, Chlamydia, Lyme dz; SE include GI upset, phlebitis)
Azithromycin (Zithromax)
Clarithromycin (Biaxin)
(used for same organisms as Erythro; also toxo & MAI; good w/ AIDS; chlamydia PID - one dose)
Ciprofloxadin (Cipro)
(cartilage damage in baby beagles)
Ofloxacin (Floxin)
(not as good for Pseudomonas)
Levofloxacin (Levaquin)
(good for gm+, QD dosing)
Moxifloxacin (Avelox)
Gatifloxacin (Tequin)
Norfloxadin (Noroxin)
(UTI and diarrhea use)
Tetracycline
Doxycycline (Vibramycin, Doryx)
Minocycline (Minocin)
Vancomycin (Vancocin)
(not absorbed PO, good for MRSA and SNA, C. diff)
Clindamycin
(bacteriostatic, not for endocarditis, not good for SNA, C. diff)
Trimethoprim-Sulfamethoxazole (Bactrim, Septra)
(for outpt UTI, OM, PCP)
Chloramphenicol (Chloromycetin)
(idiosyncratic rare irreversible aplastic anemia, dose-related toxicity causing reversible BM suppression)
Metronidazole (Flagyl)
No handout would be complete without its disclaimer… This brief summary should not replace clinical judgment. Refer to primary sources for more detailed information. Blah blah blah…

Source: http://pedicards.com/archive/antibiotics--2006.pdf

Microsoft word - global_purim

Target population: Middle school/High school students Notes: Students can work alone or in pairs, using atlases or a world map. If computers with Internet access are available, they can make use of online maps. Name: King Achashverosh was Finnish with his disobedient wife Vashti. "You Congo now!" he ordered her. After she had Ghana way, the king's messengers went Roman the land to find a

Microsoft word - v1_n1_art15.doc

QUADRO EXTENSO DE VITILIGO VULGAR DISSEMINADO EM MENOR PRÉ- Fundamento: O vitiligo é uma leucodermia adquirida relativamente frequente. Afeta 1% da população e metade dos casos inicia antes dos 20 anos. A incidência na infância é incomum. Sua causa ainda é desconhecida e a etiologia mais provável parece ser auto-imune. Objetivo: Apresentar um caso de vitiligo em menor com 3 anos, traÃ

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