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The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
November 29, 2009 (Sunday)
Registration
IUPAC Workshop
Welcome Reception
November 30, 2009 (Monday)
Opening Ceremony
Drug Discovery Research: The Synergy of Synthetic and Natural Products
Chemistry
Professor Dr. Her Royal Highness Princess Chulabhorn Mahidol
Chulabhorn Research Institute, Vipavadee-Rangsit Highway, Bangkok 10210,
Thailand.
PL-01 Exploring Synthetic Methods and Their Utilities in Enantioselective
Syntheses of Natural Products
Guo-Qiang Lin
CAS Key Laboratory of Synthetic Chemistry of Natural Substances, Shanghai
Institute of Organic Chemistry, Chinese Academy of Sciences, 345 Lingling
Road, Shanghai 200032, China.
lingq@mail.sioc.ac.cn
Poster Presentation A (Odd numbers)
Chairpersons: Zhu-Jun Yao, Prasat Kittakoop Marine Natural Products Conjuring Organic Chemistry
Takenori Kusumi, Takashi Ooi
Graduate School of Science and Engineering, Global COE Program, Tokyo
Institute of Technology, 2-12-1-H-92 Oookayama, Meguro, Tokyo 152-8551,
Japan, and Faculty of Pharmaceutical Sciences, Tokushima University,
Tokushima 770-8505, Tokushima, Japan.
kusumi.t.ab@m.titech.ac.jp
Development of Primary Amino Acid-Based Enantioselective
Organocatalytic Synthetic Methods
Xiao Han, Qiang Zhu, Jacek Kwiakowski, Zhaoqin Jiang, Lili Cheng, Xiaoyu
Wu, Jie Luo, Li-Wen Xu, Yixin Lu
Department of Chemistry, Faculty of Science & Medicinal Chemistry Program,
Life Sciences Institute, National University of Singapore, Singapore, 117543,
Republic of Singapore.
chmlyx@nus.edu.sg
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Chairpersons: Koichi Narasaka, Tony K. M. Shing PL-02 Invention of Transition Metal-Catalyzed Carbon–Carbon Bond Forming
Reactions for Organic Synthesis
Tamejiro Hiyama
Department of Material Chemistry, Kyoto University, Katsura, Nishikyo-ku,
Kyoto 615-8510, Japan.
thiyama@z06.mbox.media.kyoto-u.ac.jp
Total Syntheses of (±)-Minfiensine and (±)-Vincorine
Yong Qin
Department of Chemistry of Medicinal Natural Products, West China School
of Pharmacy, Sichuan University, Chengdu 610041, China.
yongqin@scu.edu.cn
Stereoselective Generation of (2-Fluoroalkenyl)iodonium Ylides and Their
Use for Stereoselective Synthesis of Fluoroalkenes
Shoji Hara, Satoshi Shimobaba, Guan Tong
Graduate School of Engineering, Hokkaido University, Sapporo 060-8628, Japan.
shara@eng.hokudai.ac.jp
Poster Presentation A (Even numbers)
Chairpersons: Keisuke Suzuki, Kyo Han Ahn Efficient Dye Solar Cells Based on Novel Donor-π-Acceptor Type Organic
Dyes
Tanika Khunasa, Janeeya Khunchalee, Sukrawee Pansay, Palita Kochapradit,
Siriporn Jungsuttiwng, Tinnakon Keawin, Taweesak Sudyoadsuk,
Vinich Promarak
Center for Organic Electronics and Polymers (COEP), Department of Chemistry
and Excellence Center for Innovation in Chemistry, Faculty of Science, Ubon
Ratchathani University, Warinchumrap, Ubon Ratchathani 34190, Thailand.
pvinich@sci.ubu.ac.th
Efficient Multi-Photon Excited Photoluminescence and Lasing of
π-Conjugated Oligomers
Man Shing Wong, Xin Jiang Feng, Po Lam Wu, Hoi Lam Tam, Kok Wai Cheah
Department of Chemistry and Department of Physics, Centre for Advanced
Luminescence Materials, Hong Kong Baptist University, Kowloon Tong,
Hong Kong SAR, China.
mswong@hkbu.edu.hk
Chromogenic and Fluorogenic Sensing of Heavy Metal Ions Using
Calix[4]arene Derivatives
Wen-Sheng Chung
Department of Applied Chemistry, National Chiao Tung University, Hsinchu,
Taiwan 30050.
wschung@cc.nctu.edu.tw
Business Meeting I / Dinner
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
December 1, 2009 (Tuesday)
Chairpersons: Pak Hing Leung, Toshio Nishikawa PL-03 Functional Metallopolyynes and Metallophosphors for Organic
Optoelectronics
Wai-Yeung Wong
Department of Chemistry and Centre for Advanced Luminescence Materials,
Hong Kong Baptist University, Waterloo Road, Hong Kong SAR, China.
rwywong@hkbu.edu.hk
Organic transistor/Memory Devices Based on Pentacene Films Embedding
Nanostructured Metallic or Organic Clusters
Yu-Tai Tao, Chiao-Wei Tseng
Institute of Chemistry, Academia Sinica, Taipei, Taiwan and Department of
Chemistry, National Tsing-Hua University, Hsin-Chu, Taiwan.
ytt@chem.sinica.edu.tw
Irreversible Fluorescent Chemosensors and Their Applications
Jinsung Tae, Sunho Lee, Shincheol Kang, Jihyeon Lee
Department of Chemistry, Yonsei University, Seoul 120-749, Korea.
jstae@yonsei.ac.kr
Poster Presentation B (Odd numbers)
Chairpersons: Guo-Qiang Lin, Somsak Ruchirawat The New World of Organic Chemistry in Water
Shu KobayashiDepartment of Chemistry, School of Science and Graduate School ofPharmaceutical Sciences, The University of Tokyo, Hongo, Bunkyo-ku, Tokyo113-0033, Japan.
shu_kobayashi@chem.s.u-tokyo.ac.jp Pd-Catalyzed Asymmetric Allylic Alkylation with “Hard” Carbon-
Nucleophiles
Xue-Long Hou
State Key Laboratory of Organometallic Chemistry, Shanghai Institute of
Organic Chemistry, Chinese Academy of Sciences, 354 Fenglin Lu, Shanghai
200032, China.
xlhou@mail.sioc.ac.cn
Group Picture/Lunch
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Chairpersons: Atsushi Nishida, Pauline Chiu PL-04 Development of New Stereoselective Glycosylation Methodologies and Their
Application to Oligosaccharide Synthesis
Kwan Soo Kim
Center for Bioactive Molecular Hybrids and the Department of Chemistry,
Yonsei University Seoul 120-749, Korea.
kwan@yonsei.ac.kr
Preparation of Cage-Opened Fullerene Derivatives
Liangbing Gan
Beijing National Laboratory for Molecular Sciences, Key Laboratory of
Bioorganic Chemistry and Molecular Engineering of the Ministry of Education,
College of Chemistry and Molecular Engineering, Peking University, Beijing
100871, China.
gan@pku.edu.cn
Recyclable Metal-Nanoparticle Catalysts for Organic Reactions
Jaiwook Park, Sungjin Kim, Eun Young Lee
Department of Chemistry, Pohang University of Science and Technology,
Pohang 790-784, Korea.
pjw@postech.ac.kr
Poster Presentation B (Even numbers)
Chairpersons: Chun-Chen Liao, Biing-Jiun Uang Total Synthesis of (+)-Haplophytine
Hidetoshi Tokuyama
Graduate School of Pharmaceutical Sciences, Tohoku University, Aoba 6-3,
Aramaki, Aoba-ku, Sendai 980-8578, Japan.
tokuyama@mail.pharm.tohoku.ac.jp
Multifuntional Polymeric Catalysts
Patrick H. Toy
Department of Chemistry, The University of Hong Kong, Pokfulam Road,
Hong Kong SAR, China.
phtoy@hku.hk
Total Synthesis of Natural Products: Strategies and Opportunities
David Yu-Kai Chen
Chemical Synthesis Laboratory (CSL) @ Biopolis, Institute of Chemical and
Engineering Sciences (ICES), Agency for Science, Technology and Research
(A*Star), 11 Biopolis Way, The Helios Block #03-08, Singapore 138667.
david_chen@ices.a-star.edu.sg
Excursion I (Chaopraya River Cruise)
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
December 2, 2009 (Wednesday)
Chairpersons: Sung Ho Kang, Poonsakdi Ploypradith PL-05 Synthesis of Carbocyclic Compounds through Metal-catalyzed Activation
of Alkynes
Rai-Shung Liu
Department of Chemistry, National Tsing-Hua University, Hsinchu, Taiwan.
rwywong@hkbu.edu.hk
Amidophosphane Ligand Tunable for Catalytic Asymmetric Reactions
Kiyoshi Tomioka
Synthetic Medicinal Chemistry, Graduate School of Pharmaceutical Sciences,
Kyoto University, Yoshida, Sakyo-ku, Kyoto 606-8501, Japan.
tomioka@pharm.kyoto-u.ac.jp
Asymmetric Catalysis Using Chiral N,N’-Dioxide Ligands
Xiaoming Feng
Key Laboratory of Green Chemistry & Technology, Ministry of Education,
College of Chemistry, Sichuan University, Chengdu 610064, China.
xmfeng@scu.edu.cn
Poster Presentation C (Odd numbers)
Chairpersons: Xin-Shan Ye, Hidenori Watanabe Catalytic Reactions Involving the Cleavage of C-CN Bonds
Mamaru Tobis, Naoto Chatani
Department of Applied Chemistry, Faculty of Engineering, Osaka University,
Suita, Osaka 565-0871, Japan.
chatani@chem.eng.osaka-u.ac.jp
Rediscovery of Ketene Chemistry in Different Context: Ketene-
Functionalized Polymers for Materials Application
Bongjin Moon, Minhyuck Kang, Frank Leibfarth, Craig J. Hawker
Department of Chemistry, Sogang University, Seoul 121-742, Korea and
Departments of Materials, Chemistry and Biochemistry, Materials Research
Laboratory, University of California, Santa Barbara, CA 93106, USA.
bjmoon@sogang.ac.kr
Business Meeting II
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Chairpersons: Tamejiro Hiyama, Ming-Hua Xu PL-06 Application of Organic Azides towards Synthesis of Azaheterocycles
Shunsuke ChibaDivision of Chemistry and Biological Chemistry, School of Physical andMathematical Sciences, Nanyang Technological University, Singapore 637371,Singapore.
shunsuke@ntu.edu.sg Asymmetric Synthesis with Planar Chiral Heterocycles
Katsuhiko Tomooka
Institute for Materials Chemistry and Engineering, Kyushu University,
Kasuga-koen 6-1, Kasuga-shi, Fukuoka 816-8580, Japan.
ktomooka@cm.kyushu-u.ac.jp
Poster Presentation C (Even numbers)
Chairpersons: Masahiko Yamaguchi, Keiji Tanino Pyrrolidinyl Peptide Nucleic Acids as Probes for DNA Biosensor
Applications
Cheeraporn Ananthanawat, Boonjira Boontha, Pratchayaporn Korkaew,
Voravee Hoven, Tirayut Vilaivan
Organic Synthesis Research Unit, Department of Chemistry, Faculty of Science,
Chulalongkorn University, Phayathai Road, Patumwan, Bangkok 10210, Thailand.
vtirayut@chula.ac.th
Neuritogenic Starfish Steroid Glycosides: Discovery, In Vivo Activity, and
Active Analog Synthesis
Makoto Ojika, Takayoshi, Mamiya, Yumi Sasayama, Jianhua Qi, Kouhei
Horikawa, Takuya Yagyu, Shiro Kamada, Masatoshi Haga, Youji Sakagami
Graduate School of Bioagricultural Sciences, Nagoya University, Chikusa-ku,
Nagoya 464-8601, Japan, and Faculty of Pharmacy, Meijo University,
Tenpaku-ku, Nagoya 468-8503, Japan.
ojika@agr.nagoya-u.ac.jp
Design, Synthesis and Evaluation of Iminocyclitols for the Development of
Glycosidase Inhibitors
Chun-Hung Hans Lin, Ching-Wen Ho, Yu-Rei Chuan
Institute of Biological Chemistry, Academia Sinica, No.128 Academia Road
Section 2, Nan-Kang, Taipei, 11529, Taiwan.
chunhung@gate.sinica.edu.tw
Banquet/Lectureship Award
December 3, 2009 (Thursday)
Excursion II (Grand Palace & Anatasamakhom Throne Hall)
Departure for the Suvannabhumi International Airport
Return to the Residence/The Miracle Grand Hotel
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
POSTER PRESENTATION
November 30, 2009 (Monday)
Poster Presentation Session A
Annulation–Cyclization Approach to Polyketide-Derived Polycyclic Natural Products
Keisuke Suzuki
Department of Chemistry, Tokyo Institute of Technology, SORST–JST, 2-12-1, O-okayama,
Meguro-ku, Tokyo 152-8551, Japan.
ksuzuki@chem.titech.ac.jp
Asymmetric Synthesis of Chiral Pyroglutamates and Their Application in the Synthesis
of Pyrrolizidine Alkaloids
Chuan-Chung Chung, Kwan-Wen Lin, Yen-Fang Wen, Yi-Fang Lin, Biing-Jiun Uang
Department of Chemistry, National Tsing Hua University, Hsinchu, Taiwan 30013.
bjuang@mx.nthu.edu.tw
Total Synthesis of Crinipellin B
Wonyeob Kim, Mi-Hee Han, Seog-Bum Song, Hee-Yoon Lee
Department of Chemistry, Korea Advanced Institute of Science and Technology, Daejeon
305-701, Korea.
leehy@kaist.ac.kr
Intramolecular Direct Aldol Reactions of Sugar Diketones
Tony K. M. Shing, Hau M. Cheng
Department of Chemistry and Center of Novel Functional Molecules, The Chinese University
of Hong Kong, Shatin, Hong Kong SAR, China.
tonyshing@cuhk.edu.hk
A Novel Reverse Prenylation of Indole Derivatives by Means of Acetylene Cobalt Complex
Toshio Nishikawa, Hisaaki Isaji, Atsuo Nakazaki, Minoru Isobe
Graduate School of Bioagricultural Sciences, Nagoya University, Chikusa, Nagoya 464-8601,
Japan and Department of Chemistry, National Tsing Hua University, Hsinchu 300131, Taiwan.
nisikawa@agr.nagoya-u.ac.jp
“On water” Mediated Reaction of Nitroolefins with Various Nucleophiles
Ching-Fa Yao
Department of Chemistry, National Taiwan Normal University, 88, Sec. 4, Tingchow Road,
Taipei 116, Taiwan.
cheyaocf@ntnu.edu.tw
Total Synthesis of Polyanthellin A on the Basis of a Higher Order Cycloaddition Reaction
Keiji Tanino, Koichiro Dota
Faculty of Science, Hokkaido University, Sapporo 060-0810 Japan.
ktanino@sci.hokudai.ac.jp
Friedel Crafts Arylations
Simon Duttwyler, Anthony Linden, Kim K. Baldridge, Jay S. Siegel
Organic Chemistry Institute, University of Zurich, Winterthurerstrasse 190, Zurich 8057,Switzerland.
jss@oci.uzh.ch The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Synthesis and Biological Activities of Azalamellarins
Nopporn Thasana, Sasiwadee Boonya-udtayan, Nattawut Yotapan, Carson Bruns, Christina
Woo, Somsak Ruchirawat
Laboratory of Medicinal Chemistry, Chulabhorn Research Institute, and Program in Chemical
Biology, Center for Environmental Health, Toxicology and Management of Toxic Chemicals,
Chulabhorn Graduate Institute, Vipavadee-Rangsit Highway, Bangkok 10210 Thailand.
nopporn@cri.or.th
A Novel Total Synthesis of Estrone
Wei-Dong Z. Li, Ya-Ping Xue
State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou 730000
and State Key Laboratory & Institute of Elemento-organic Chemistry, Nankai University,
Tianjin 300071, China.
wdli@nankai.edu.cn
A New Approach towards 6-Membered Azacycles Using Gold(I)-Catalyzed
Cycloisomerization of Mixed N,O-Acetals
Young Ho Rhee, Cheoljae Kim, Hyo Jin Bae, Haejin Kim, Vasu Sampath
Department of Chemistry, POSTECH (Pohang University of Science and Technology),
Hyoja-dong San 31, Pohang, Kyungbook, Republic of Korea, 790-784.
yhrhee@postech.ac.kr
Intramolecular Nucleophilic Addition Reactions of Tertiary Enamides to Epoxides and
Ketones, Highly Efficient and Selective Approaches to Clausena Alkaloids and Analogs
Luo Yang, De-Xian Wang, Zhi-Tang Huang, Mei-Xiang Wang
National Laboratory for Molecular Sciences, CAS Laboratory of Molecular Recognition and
Function, Institute of Chemistry, Chinese Academy of Sciences, Beijing 100190, China, and
The Key Laboratory of Bioorganic Phosphorus Chemistry & Chemical Biology (Ministry of
Education), Department of Chemistry, Tsinghua University, Beijing 100084, China.
wangmx@mail.tsinghua.edu.cn, mxwang@iccas.ac.cn
Synthetic study of Unexpected C-Aminoglycosylation via Barbier-Grignard Type
Allylation/Propargylation of Glycal: An Approach to Sialic Acids
Rujee Lorpitthaya, Siming Wang, Kalyan Kumar Pasunooti, Xiaozhou Luo, Xue-Wei Liu
Division of Chemistry and Biological Chemistry, School of Physical and Mathematical
Sciences, Nanyang Technological University, Singapore 637313.
xuewei@ntu.edu.sg
Disulfides Exchange Reaction of Insulin Using Rhodium Trichloride
Mieko Arisawa, Manabu Kuwajima, Masahiko Yamaguchi
Department of Organic Chemistry, Graduate School of Pharmaceutical Sciences, WPI
Advanced Institute for Materials Research, Tohoku University, Aoba, Sendai 980-8577, Japan.
yama@mail.pharm.tohoku.ac.jp
Sequential One Pot Synthesis of Dibenzo[a,c]cyclohepten-5-ones and Their Biological
Activities Against Cancer Cell Lines
Poolsak Sahakitpichan, Juthatip Boonsombat, Somsak Ruchirawat
Laboratory of Natural Products, Chulabhorn Research Institute, and Program in Chemical
Biology, Chulabhorn Graduate Institute, Vipavadee-Rangsit Highway, Bangkok 10210,
Thailand.
poolsak@cri.or.th
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Novel Asymmetric Domino Reactions Promoted by Acid-Base Organocatalysts
Shinobu Takizawa, Naohito Inoue, Hiroaki Sasai
The Institute of Scientific and Industrial Research (ISIR), Osaka University, Mihogaoka,
Ibaraki-shi, Osaka 567-0047, Japan.
sasai@sanken.osaka-u.ac.jp
Non-classical Bonding in Carbon Chemistry: Bent Allenes, Carbenes, Zwitterions or
Carbon(0)-Complexes?
Han Vinh Huynh, Yuan Han, Li Juan Lee
Department of Chemistry, National University of Singapore, 3 Science Drive 3, 117543
Singapore.
chmhhv@nus.edu.sg
Development of New Direct Catalytic Reactions Using Tetranuclear Zinc Clusters
Takashi Ohshima, Takanori Iwasaki, Yusuke Maegawa, Yukiko Hayashi, Kazushi Agura,
Kazushi Mashima
Department of Chemistry, Graduate School of Engineering Science, Osaka University 1-3
Machikaneyama, Toyonaka, Osaka 560-8531, Japan.
ohshima@chem.es.osaka-u.ac.jp
Formal Total Synthesis of N-Methylmaysenine
Zhen Yang
College of Chemistry and Molecular Engineering, Peking University, Beijing 100871, China
and Laboratory of Chemical Genomics, School of Chemical Biology and Biotechnology,
Shenzhen Graduate School of Peking University, Shenzhen 518055, China.
zyang@pku.edu.cn
Asymmetric Diels-Alder Reaction of Danishefsky Dienes
Atsushi Nishida, Shinji Harada, Siharu Hiraoka, Nozomi Toudou, Daisuke Shirasaki,
Yukinori Sudo
School of Pharmaceutical Sciences, Chiba University, 1-33 Yayoi-cho, Inage-ku, Chiba
263-8522, Japan.
nishida@p.chiba-u.ac.jp
Synthesis of gem-Difluoromethylenated 1-Azabicyclic Compounds by Fluoride-Catalyzed
Addition of PhSCF SiMe to N-Substituted Cyclic Imides Followed by Radical Cyclization
Manat Pohmakotr, Teerawut Bootwicha, Duanghathai Panichakul, Chutima Kuhakarn,Samran Prabpai, Palangpon Kongsaeree, Patoomratana Tuchinda, Vichai ReutrakulDepartment of Chemistry and Center for Innovation in Chemistry, Faculty of Science,Mahidol University, Rama VI Road, Bangkok 10400, Thailand.
scmpk@mahidol.ac.th Total Synthesis of Bioactive Natural Alkaloid Maistemonine
Yong-Qiang Tu
State Key Laboratory of Applied Organic Chemistry, Department of Chemistry,
Lanzhou University, Lanzhou 730000, China.
tuyq@lzu.edu.cn
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Bioactive Compounds from Thai Fungi
Porntep Chomcheon, Nattha Ingavat, Suthep Wiyakrutta, Nongluksna Sriubolmas, Nattaya
Ngamrojanavanich, Chulabhorn Mahidol, Somsak Ruchirawat, Prasat Kittakoop
Chulabhorn Research Institute, Vibhavadi Rangsit Road, Bangkok 10210, Thailand, Program
of Biotechnology, Chulalongkorn University, Chulabhorn Graduate Institute, Department of
Microbiology, Mahidol University, Department of Microbiology, Chulalongkorn University,
and Chulabhorn Research Centre, Institute of Science and Technology for Research and
Development, Mahidol University, Thailand.
prasat@cri.or.th
Programmable Assembly of Metal Complexes
Kentaro Tanaka, Yasuyuki Yamada, Shin-ichiro Kawano, Yusuke Takezawa, Guido H. Clever,
Mitsuhiko Shionoya
Department of Chemistry, Graduate School of Science, Nagoya University, Furo-cho, Chikusa-
ku, Nagoya 464-8602, Japan, and Department of Chemistry, Graduate School of Science,
The Universityof Tokyo, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.
kentaro@chem.nagoya-u.ac.jp
Antibacterial Metabolites from the Endophytic Fungi of the Genus Botryosphaeria
Vatcharin Rukachaisirikul, Wipapan Pongcharoen, Jiraporn Arunpanichlert, Yaowapa
Sukpondma, Souwalak Phongpaichit, and Jariya Sakayaroj
Department of Chemistry and Center for Innovation in Chemistry, Department of Microbiology,
Faculty of Science, Prince of Songkla University, Hat Yai, Songkhla 90112, Thailand, and
National Center for Genetic Engineering and Biotechnology, Thailand Science Park, Klong
Luang, Pathumthani, 12120, Thailand.
vatcharin.r@psu.ac.th
New Indoles and Benzo[b]furans as Electroluminescent Materials
Jih Ru Hwu, Yung Chang Hsu, Kao-Shuh Chuang, Thainashmuthu Josephrajan, Shwu-Chen Tsay
Department of Chemistry, National Central University, Jhongli, Taiwan 32001, and Department
of Chemistry, National Tsing Hua University, Hsinchu, Taiwan 30013.
jrhwu@mx.nthu.edu.tw
Development of “Turn-On” Fluorescent Probes for Amino-Carboxylates and Metal Ions
Based on Organic Reactions
Kyo Han Ahn, Dowook Ryu, Amrita Chatterjee, Mithun Santra
Department of Chemistry and Center for Electro-Photo Behaviors in Advanced Molecular
Systems, POSTECH, San 31 Hyoja-dong, Pohang, 790-784, Korea.
ahn@postech.ac.kr
Preparation and Fluorescence Characterization of Selected Derivatives of Quinoxaline,
Quinoline and Benzoimidazole
Hairul Anuar Tajuddin, Zanariah Abdullah, Noor Doha Hassan, Zainal Abidin Hasan
Department of Chemistry, Faculty of Science, University of Malaya, 50603 Kuala Lumpur, Malaysia.
hairul@um.edu.my
Engineering of Protein-Based Biosensor for Sensing of Metal Ion and Reactive Oxygen Species
Chartchalerm Isarankura-Na-Ayudhya, Tanawut Tantimongcolwat, Virapong Prachayasittikul
Department of Clinical Microbiology, Faculty of Medical Technology, Mahidol University,
Bangkok 10700 Thailand.
mtcis@mahidol.ac.th
Towards Controlling Self Organization of Discotic Liquid Crystal: Overcoming Core
Dipole Interaction by Rational Design of Amphiphilic Peripheral Side Chains
Yu-Lou Su, Mei-Chin Tzeng, Chi Wi Ong
Department of Chemistry, National Sun Yat Sen University, Kaoshiung, Taiwan 804.
cong@mail.nsysu.edu.tw
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Highly Efficient Asymmetric Polar Head Cholesterol-Based Cationic Lipids for DNA
Delivery to Human Prostate Adenocarcinoma Cells
Boon-ek Yingyongnarongkul, Widchaya Radchatawedchakoon, Aungkana Krajarng, Ramida
Watanapokasin, Apichart Suksamrarn
Department of Chemistry, Faculty of Science, Ramkhamhaeng University, Bangkapi, Bangkok
10240, Thailand, and Department of Biochemistry, Faculty of Medicine, Srinakharinwirot
University, Wadhana, Bangkok 10110, Thailand.
boonek@ru.ac.th
Marine Polycyclic Ethers-Molecular Mode of Action
Tohru Oishi, Satoru Ujihara, Kohei Torikai, Nobuaki Matsumori, Michio Murata
Department of Chemistry, Osaka University, 1-1 Machinakeyama, Toyonaka, Osaka 560-0043,
Japan.
murata@ch.wani.osaka-u.ac.jp
The Novel Antimetastatic Agents: A Breakthrough in the Treatment of Lung and Breast
Cancers
Wen-Shan Li, Kai-Hsuan Chang, Tzu Ting Chang, Ya Ching Jen, Kung-Cheng Liu, Chin-
Chun Hung,Yi-Ching Wang, Wen-Chun Hung, Shu-Chuan Jao
Institute of Chemistry, Academia Sinica, Department of Pharmacology, National Cheng Kung
University, Institute of Biomedical Sciences, National Sun Yat-Sen University, and Institute
of Biological Chemistry, Academia Sinica, Taipei, Taiwan.
wenshan@gate.sinica.edu.tw
Development of a Set of Simple, Interpretable ADMET Rules of Thumb
M. Paul Gleeson
Kasetsart University, Department of Chemistry, Faculty of Science, 50 Phaholyothin Rd,
Chatuchak, Bangkok 10900, Thailand, and Chulabhorn Research Institute, Laboratory of
Medicinal Chemistry, Vipavadee-Rangsit Highway, Bangkok 10210 Thailand.
paul.gleeson@ku.ac.th
High Performances of Gold Nano-particles Supported on Cobalt Oxide (Au/Co O ) as
an Alternative Catalyst for Homogeneous Cobalt Carbonyls
Makoto Tokunaga, Akiyuki Hamasaki, Xiaohao Liu, Yoshihiro Yamane, Shingo Haraguchi
Department of Chemistry, Kyushu University, 6-10-1 Hakozaki, Higashi-ku, Fukuoka
812-8581, Japan.
mtok@chem.kyushu-univ.jp
An Indolocarbazole Oligomer Binding Sulfate Ion with High Selectivity and Its Crystal
Structure of Helical Conformation
Kyu-Sung Jeong, Jun-il Kim
Center for Bioactive Molecular Hybrids, Department of Chemistry, Yonsei University Seoul,
120-749, Korea.
ksjeong@yonsei.ac.kr
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
December 1, 2009 (Tuesday)
Poster Presentation Session B
Synthesis of Symmetrical and Unsymmetrical N-Aryl and N-Alkyl Ureas and Recent
Advances on C-N coupling
Man-kit Leung
Department of Chemistry and Institute of Polymeric Science and Engineering, National Taiwan
University, 1 Roosevelt Road, Sec. 4, Taipei, Taiwan.
mkleung@ntu.edu.tw
Palladium-Catalyzed Annulation of 2-(1-Alkynyl)biphenyls with Aryl Iodides to Di-
substituted Methylidenefluorenes
Chin-Chau Chen, Shyh-Chyun Yang, Ming-Jung Wu
School of Pharmacy, Kaohsiung Medical University, Kaohsiung, Taiwan, and Department of
Chemistry, National Sun Yat-sen University, Kaohsiung, Taiwan.
mijuwu@faculty.nsysu.edu.tw
Stereoselective Three Component Coupling Reaction for beta-Branched Morita-Baylis-
Hillman Ester
Do Hyun Ryu, Sung Il Lee, Bidyut Kumar Senapati, Geum-Sook Hwang
Department of Chemistry, Sungkyunkwan University, Suwon 440-746 and Korea Basic Science
Institute, 5St, Anam-Dong, Seongbuk-Gu, Seoul, Korea.
dhryu@skku.edu
Synthesis and Evaluation of Novel Non-peptide Corticotropin Releasing Hormone
Receptor-1 Antagonists for Imaging Studies
B. Moon Kim, Chiyeun Chough, Jin Kyu Choi
Department of Chemistry, College of Natural Sciences, Seoul National University, Seoul,
151-747, Korea.
kimbm@snu.ac.kr
Allene Cyclisations for Heterocycle Synthesis
Roderick W. Bates, M. R. Dewey, C. J. Lim, Y. Lu, S. Sridhar
Division of Chemistry and Biological Chemistry, School of Physical and Mathematical
Sciences, Nanyang technological University, 21 Nanyang Link, Singapore 637371.
Roderick@ntu.edu.sg
Polymer-Supported N-Phenylsulfonyloxaziridine (Davis Reagent): A Versatile Oxidant
Yulin Lam, Yongnian Gao
Department of Chemistry, National University of Singapore, 3 Science Drive 3, Singapore
117543.
chmlamyl@nus.edu.sg
Expeditious Access to Natural Product Analogs Employing Versatile Scaffolds: Systematic
Diversification of Ring-junctions and Divergent Cyclizations
Hiroki Oguri, Takahisa Hiruma, Haruki Mizoguchi, Hideaki Oikawa
Division of Chemistry, Graduate School of Science, and Division of Innovative Research,
Creative Research Initiative ‘Sousei’ (CRIS), Hokkaido University, Japan.
oguri@sci.hokudai.ac.jp
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Aluminum-Mediated Direct Carboxylation of Aromatic Compounds with CO2
–Applicability and Dichotomy of the Reaction Mechanism–
Tetsutaro Hattori, Koji Nemoto, Satoru Onozawa, Naoya Morohashi
Department of Environmental Studies, Graduate School of Environmental Studies, Tohoku
University, 6-6-11 Aramaki-Aoba, Aoba-ku, Sendai 980-8579, Japan.
hattori@orgsynth.che.tohoku.ac.jp
Synthetic Studies toward Marine Alkaloid (–)-Nakadomarin A
Bin Cheng, Hongbin Zhai
The Key Laboratory of Synthetic Chemistry of Natural Substances, Shanghai Institute of Organic
Chemistry, Chinese Academy of Sciences, Shanghai 200032, China and The State Key
Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing 100083, China.
zhaih@mail.sioc.ac.cn
Efficient Total Synthesis of Water Soluble (S)-14-Azacamptothecin
Zhu-Jun Yao, Guan-Sai Liu
State Key Laboratory of Bioorganic and Natural Products Chemistry, Shanghai Institute of
Organic Chemistry, Chinese Academy of Sciences, 345 Lingling Road, Shanghai 200032,
China, and Nanjing National Laboratory of Microstructures, School of Chemistry and Chemical
Engineering, Nanjing University, 22 Hankou Road, Nanjing 210093, China.
yaoz@mail.sioc.ac.cn, yaoz@nju.edu.cn
Chemical Transformation of the Cinchona Alkaloid
Didin Mujahidin, Maria Mardiastuti, Hans M. Rudolf Hoffmann
Division of Organic Chemistry, Faculty of Mathematics and Natural Sciences, Institut Teknologi
Bandung, Jalan Ganesa 10, Bandung 40132, Indonesia. Fax. 62-22-2504154, and Department
of Organic Chemistry, University of Hannover, Schneinberg 1 B, Hannover 30176, Germany.
didin@chem.itb.ac.id
Ortho-Quinone Methides Generated by p-TsOH on Silica and Their [4+2]-Cycloaddition
Reactions with Styrenes
Poonsakdi Ploypradith, Jumreang Thummatorn, Paratchata Batsomboon, Suttipol Radomkit,
Somsak Ruchirawat
Laboratory of Medicinal Chemistry, Chulabhorn Research Institute, and Program in Chemical
Biology, Chulabhorn Graduate Institute, Vipavadee-Rangsit Highway, Bangkok 10210,
Thailand.
poonsakdi@cri.or.th
A New Method for Synthesis of 2-Deoxyglycosides from D-glucal by Using Iodine
Monobromide
Rungnapha Saeeng, Uthaiwan Sirion, Pornhathai Kankaew
Department of Chemistry and Center for Innovation in Chemistry, Faculty of Science, Burapha
University, Sangsook, Chonburi 20131, Thailand.
rungnaph@buu.ac.th
Nitrones: An Expeditious Access to 1-Aminoindanes
Hyun-Suk Yeom, Youngun Lee, Jaewon Jeong, Seunghoon Shin
Department of Chemistry, Hanyang University, Seoul, Korea, 133-791.
sshin@hanyang.ac.kr
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Synthetic Studies on (–)-Gelsemoxonine
Jun Shimokawa, Satoshi Yokoshima, Tohru Fukuyama
Laboratory of Synthetic Natural Products Chemistry, Graduate School of Pharmaceutical
Sciences, University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.
jshimok@mol.f.u-tokyo.ac.jp
Spectroscopic Analyses and Chemical Transformations for Structure Elucidation of Novel
Indole Alkaloids from Gelsemium elegans
Noriyuki Kogure, Yousuke Yamada, Mariko Kitajima, Sumphan Wongseripipatana,
Hiromitsu Takayama
Graduate School of Pharmaceutical Sciences, Chiba University, Chiba 263-8522, Japan.
nkogure@p.chiba-u.ac.jp
Stereoselective Synthesis of Aryl 2-Deoxy-C-glycosides by Palladium-Catalyzed Coupling
Reactions
Xin-Shan Ye, De-Cai Xiong, Hou-Hua Li
State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences,
Peking University, Xue Yuan Road No. 38, Beijing 100191, China.
xinshan@bjmu.edu.cn
Tetrahydro-1,4-epoxynaphthalene-1-carboxylic acid: A New Chiral Derivatizing Agent
for Determination of the Absolute Configuration of Secondary Alcohols
Suttipun Sungsuwan, Nopporn Ruangsupapichart, Tienthong Thongpanchang
Department of Chemistry and Center for Innovation in Chemistry, Faculty of Science, Mahidol
University, Rama 6 Road, Bangkok 10400 Thailand, and National Center for Genetic
Engineering and Biotechnology, Thailand Science Park, Klong Luang, Patumthani 12130,
Thailand.
tettp@mahidol.ac.th
AminoOrganoBoron (AOB) Complexes for Molecular Catalysis: Control of Hydrogen
Transfer Process in Organic Synthesis
Shunsuke Oishi, Junichi Yoshimoto, Ryoji Noyori, Susumu Saito
Graduate School of Science & Institute for Advanced Research, Nagoya University, Chikusa,
Nagoya, 464-8602, Japan.
saito.susumu@f.mbox.nagoya-u.ac.jp
Suzuki-Miyaura Coupling of Alkyl Halides Catalyzed by Novel Iron-Phosphine Complexes
Masaharu Nakamura
International Research Center for Elements Science, Institute for Chemical Research, Kyoto
University, Uji, Kyoto, 611-0011, Japan.
masaharu@scl.kyoto-u.ac.jp
Enantioselective Oxidative Kinetic Resolution of Racemic Secondary Alcohols Using
Chirally Modified AZADOs
Yoshiharu Iwabuchi
Graduate School of Pharmaceutical Sciences, Tohoku University, 6-3 Aobayama, Sendai 980-
8578, Japan.
iwabuchi@mail.pharm.tohoku.ac.jp
Biologically Active Prenylated Flavonoids from the Roots of Eriosema chinense
Somyote Sutthivaiyakit, Oracha Thongnak, Thitima Lhinhatrakool, Orapan Yodchun, Ratree
Srimark, Prisana Dowtaisong, and Mayuree Chuankamnerdkarn
Department of Chemistry and Center for Innovation in Chemistry, Faculty of Science,
Ramkhamhaeng University, Hua Mark, Bangkapi, Bangkok 10240, Thailand.
s_somyote@ru.ac.th
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Bioactive Ingredients from the Mangrove and Thai Medicinal Plants
Chatchanok Karalai, Chanita Ponglimanont, Suchada Chantrapromma, Akkharawit Kanjana-
Opas, Supinya Tiewtrakul, Kan Chantrapromma, Hoong Kun-Fun
Department of Chemistry, Faculty of Science, Prince of Songkla University, Hat-Yai, Songkhla
90110, Thailand.
chatchanok.k@psu.ac.th
Computational Modeling of Imprinting Factor of Molecularly Imprinted Polymers via
Data Mining Approach
Chanin Nantasenamat, Chartchalerm Isarankura-Na-Ayudhya, Virapong Prachayasittikul
Department of Clinical Microbiology, Faculty of Medical Technology, Mahidol University,
Bangkok 10700, Thailand.
mtcnt@mahidol.ac.th
A New Bipolar Material for Highly Efficient Deep-Blue Fluorescence, Yellow-Green
Phosphorescence and White OLEDs
Ken-Tsung Wong
Department of Chemistry, National Taiwan University, Taipei 10617, Taiwan.
kenwong@ntu.edu.tw
Chromogenic and Fluorogenic Sensing of Cu2+ based on Thiazole Derivatives
Hong-Seok Kim, Aasif Helal, Sang Hoon Lee, Sang Hyun Kim
Department of Applied Chemistry, Kyungpook National University, Daegu, 702-701, Korea.
kimhs@knu.ac.kr
Reversible Switching Between Hydrophilic and Hydrophobic Magnetic Microsphere
Surfaces via One-Step Supramolecular Dynamic Dendronization
Ken Cham-Fai Leung, Shouhu Xuan
Center of Novel Functional Molecules, Department of Chemistry, The Chinese University of
Hong Kong, Shatin, NT, Hong Kong SAR, China.
cfleung@cuhk.edu.hk
Bisanthene-based Soluble and Stable Near-Infrared Dyes
Kai Zhang, Junhong Yao, Jinling Li, Jishan Wu
Department of Chemistry, National University of Singapore, 3 Science Drive 3, 117543,
Singapore.
chmwuj@nus.edu.sg
Confusion Approach to Near-IR Luminescent Porphyrinoids
Hiroyuki Furuta
Department of Chemistry and Biochemistry, Graduate School of Engineering, Kyushu
University, Fukuoka 819-0395, Japan.
hfuruta@cstf.kyushu-u.ac.jp
Cereulide, an Emetic Toxin from B. cereus Takes Antipodal Frame with Different Chem-
bio-activities from Valinomycin, an Antibiotic from S. fulvissimus
Minoru Isobe, Arthit Makarasen
Chemistry Department, National Tsing Hua University, 101 Sec. 2, Kuang Fu Road, Hsinchu
30013 Taiwan, and Chulabhorn Research Institute, Vipavadee-Rangsit Highway, Bangkok
10210, Thailand.
minoru@mx.nthu.edu.tw
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Biosynthetic Studies of Macrolide Antibiotic FD-891 Produced by Streptomyces
graminofaciens A-8890
Fumitaka Kudo, Atsushi Motegi, Akiko Komatsubara, Tadashi Eguchi
Department of Chemistry, Graduate School of Science and Engineering, Tokyo Institute of
Technology, 2-12-1 O-okayama, Meguro-ku, Tokyo 152-8551, Japan.
fkudo@chem.titech.ac.jp
Synthesis of Natural Product-like Compounds with Anti-tumor Bioactivities
Jingbo Chen, Zhuxian Sun, Xianghui Zeng, Jianping Liu, Liang Li, Hongbin Zhang
Key Laboratory of Medicinal Chemistry for Natural Resource, Ministry of Education, School
of Chemical Science and Technology, Yunnan University, Kunming, Yunnan 650091, China.
zhanghb@ynu.edu.cn
Evaluation of the Anti-inflammatory Potential of Tectona grandis
Christine L. Chichioco-Hernandez, Noemi D. Paguigan, Jeffrey D. de Vera
Institute of Chemistry, College of Science, University of the Philippines, Diliman, Quezon
City 1101, Philippines.
cchernandez@up.edu.ph
Structural Modification of Lamellarins to Optimize Their Cytotoxic Activities and Drug-
like Properties
Montakarn Chittchang, M. Paul Gleeson, Poonsakdi Ploypradith, Somsak Ruchirawat
Laboratory of Medicinal Chemistry, Chulabhorn Research Institute, and Chemical Biology
Program, Chulabhorn Graduate Institute, Vibhavadee-Rangsit Highway, Bangkok 10210,
Thailand, and Department of Chemistry, Faculty of Science, Kasetsart University, Phaholyothin
Road, Chatuchak, Bangkok 10900, Thailand.
montakarn@cri.or.th
Investigation of Antioxidative and Antimicrobial Activities of 1-Adamantylthio analog
of Pyridines and Tetrahydropyridines
Supaluk Prachayasittikul, Lertyot Treeratanapiboon, Ratana Lawung, Ratchanok Pingaew,
Apilak Worachartcheewan, Somsak Ruchirawat, Virapong Prachayasittikul
Department of Chemistry, Faculty of Science, Srinakharinwirot University, Bangkok
10110,Thailand, Department of Parasitology, Faculty of Medical Technology, Mahidol
University, Bangkok 10700, Thailand, Department of Clinical Microbiology, Faculty of
Medical Technology, Mahidol University, Bangkok 10700, Thailand, and Laboratory of
Medicinal Chemistry, Chulabhorn Research Institute, Bangkok 10210, Thailand.
supaluk@swu.ac.th
Hydrogen-bonding-mediated Supramolecular Porphyrin Array
Woo-Dong Jang, Dongyong Kim, Jungmi Heo, Chi-Hwa Lee
Department of Chemistry, College of Science, Yonsei University, 262 Seongsanno,
Seodaemun-gu, Seoul 120-749, Korea.
wdjang@yonsei.ac.kr
Isomerization Polymerization of Cycloolefins Catalyzed by Pd Complexes. Synthesis of
Liquid Crystalline Hydrocarbon Polymers
Kohtaro Osakada, Daisuke Takeuchi, Park Sehoon, Takeshi Okada
Chemical Resources Laboratory R1-03, Tokyo Institute of Technology, 4259 Nagatsuta,
Midori-ku, Yokohama, 226-8503, Japan.
kosakada@res.titech.ac.jp
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
December 2, 2009 (Wednesday)
Poster Presentation Session C
Photooxygenation of Masked o-Benzoquinones: An Efficient Entry to Highly
Functionalized Cyclopentenones from 2-Methoxyphenols
Tzu-Chiao Kao, Chun-Chen Liao
Department of Chemistry, National Tsing Hua University, Hsinchu, Taiwan 30013, and
Department of Chemistry, Chung-Yuan Christian University, Taoyuan, Taiwan 32023.
ccliao@cycu.edu.tw
Total Synthesis of Azithromycin
Hyoung Cheul Kim, Sung Ho Kang
Department of Chemistry, KAIST, Daejeon 305-701, Korea.
shkang@kaist.ac.kr
Natural Products Synthesis from Chiral Aziridine-2-carboxylates
Yongeun Kim, Hee-Sung Eum, Alok Singh, Hyun-Joon Ha
Department of Chemistry, Hankuk University of Foreign Studies, Yongin, 449-791, Korea.
hjha@hufs.ac.kr
Copper-mediated Reductions of Unsaturated Thioesters
Ninglin Li, Pauline Chiu
Department of Chemistry and Open Laboratory of Chemical Biology of the Institute of
Molecular Technology for Drug Discovery and Synthesis, University of Hong Kong,
Pokfulam Rd., Hong Kong SAR, China.
pchiu@hku.hk
Palladium-Catalyzed Direct Cross-Coupling of Olefins with Acrylates
Teck Peng Loh
Division of Chemistry and Biological Chemistry, School of Physical and Mathematical
Sciences, Nanyang Technological University, Singapore 637371, Singapore.
teckpeng@ntu.edu.sg
Catalytic Electron Transfer Reaction for Organic Synthesis: Cyclization of Alkenyl and
Alkynyl N-Benzoyloxysulfonamides to Pyrrolidine Derivatives
Wei-Min Liu, Zheng-Hong Liu, Koichi Narasaka
Division of Chemistry and Biological Chemistry, School of Physical and Mathematical
Sciences, Nanyang Technological University, SPMS-04-01, 21 Nanyang Link, Singapore
637371, Singapore.
narasaka@ntu.edu.sg
Asymmetric Approach to the Pentacyclic Skeleton of Aspidosperma Alkaloids via
1,3-Dipolar Cycloaddition of Carbonyl Ylides Catalyzed by Chiral Rh(II) Complexes
Hisanori Nambu, Mayuka Hikime, Megumi Kamiya, Naoyuki Shimada, Shunichi Hashimoto
Faculty of Pharmaceutical Sciences, Hokkaido University, Sapporo 060-0812, Japan.
nambu@pharm.hokudai.ac.jp
Gold-Catalyzed Functionalization of Silyl Enol Ethers
Naoki Asao, Haruo Aikawa, Tetsuro Kaneko
Department of Chemistry, Graduate School of Science, Tohoku University, Sendai 980-8578,
Japan.
asao@m.tains.tohoku.ac.jp
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Exploring Chiral Vicinal Diamines as Highly Effective Ligands for Transition Metal
Catalysis: Asymmetric Synthesis of Enantioenriched Phthalides
Ming-Hua Xu, Shen-Shuang Jin, Bo Zhang, Chun Shen, Bao-Jian Pei, Guo-Qiang Lin
Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road,
Shanghai 201203, and Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences,
345 Lingling Road, Shanghai 200032, China.
xumh@mail.sioc.ac.cn
Enantioselective Total Syntheses of Marine Natural Products Awajanomycin and
Ypaoamide
Jie Chen, Rui Fu, Pei-Qiang Huang
Department of Chemistry and Key Laboratory for Chemical Biology of Fujian Province,
College of Chemistry and Chemical Engineering, Xiamen University, Xiamen 361005, China.
pqhuang@xmu.edu.cn
New Method for Stereo- and Regioselective Synthesis of The 4-Halogeno (Cl-, Br-)-Pregn-
4-en-16α-ol-17α-fluo-3-on-20-yne, New Ethynylsteroidal Substance Class
Luu Duc Huy
Laboratory of Steroids & Alkaloids, Institute of Chemistry, Vietnamese Academy of Science
and Technology, 18 Hoang Quoc Viet, Hanoi, Vietnam.
ldhuy@netnam.vn
New Synthetic Applications of o-Iodoxybenzoic Acid (IBX) in Organic Synthesis
Chutima Kuhakarn, Supanimit Chiampanichayakul, Waraporn Panchan, Manat Pohmakotr,
Vichai Reutrakul, Thaworn Jaipetch
Department of Chemistry and Center for Innovation in Chemistry, Faculty of Science,
Mahidol University, Rama VI Road, Bangkok 10400, Thailand.
scckk@mahidol.ac.th
Progess in the Synthesis and Cytotoxicity of Tylophora Alkaloids
Wannaporn Disadee, Somsak Ruchirawat
Laboratory of Medicinal Chemistry, Chulabhorn Research Institute, and Program in Chemical
Biology, Chulabhorn Graduate Institute, Vipavadee-Rangsit Highway, Bangkok 10210,
Thailand.
wannapor@cri.or.th
Switchable Reactivity of b–Keto Esters Toward Alkenes and Modulated Selective
Synthesis of O-Heterocycles and Carbocycles by Tuning Metal Catalysts
So Won Youn
Department of Chemistry, Pukyong National University, Busan 608-737, Korea.
sowony@pknu.ac.kr
Synthetic Study on Solanoeclepin A
Hidenori Watanabe, Yusuke Nakatani, Yoshifumi Kusumoto, Tadashi Imaoka
Department of Applied Biological Chemistry, Graduate School of Agricultural and Life
Sciences, the University of Tokyo 1-1-1 Yayoi, Bunkyo-ku, Tokyo 113-8657, Japan.
ashuten@mail.ecc.u-tokyo.ac
Palladium-Catalyzed C-C Bond Formations Using Phosphine-Free Hydrazone Ligands
Takashi Mino, Kenji Kajiwara, Tomoko Koizumi, Masami Sakamoto, Tsutomu Fujita
Department of Applied Chemistry and Biotechnology, Graduate School of Engineering, Chiba
University, Chiba, 263-8522, Japan.
tmino@faculty.chiba-u.jp
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Asymmetric Organocatalyzed Relay Cascades: Efficient Protocol for Constructing
Complex Molecules Containing Multiple Stereocentres
Yao Wang, Peng-Fei Xu
State Key Laboratory of Applied Organic Chemistry, College of Chemistry and Chemical
Engineering, Lanzhou University, Lanzhou 730000, China.
xupf@lzu.edu.cn
Synthesis and Screening for Acetylcholinesterase Inhibitory Activity of Some Novel
Coumarin Derivatives
Dumrongsak Aryuwananon, Nisachon Khunnawutmanotham, Nitirat Chimnoi, Kornkanok
Ingkaninan, Supanna Techasakul
Department of Chemistry and Center for Innovation in Chemistry, Faculty of Science, Kasetsart
University, Jatujak, Bangkok 10900, Thailand, Chulabhorn Research Institute, Vibhavadee-
Rangsit Road, Laksi, Bangkok 10210, Thailand, and Department of Pharmaceutical Chemistry
and Pharmacognosy, Faculty of Pharmaceutical Sciences, Naresuan University, Phitsanulok
65000, Thailand.
fscispt@ku.ac.th
Structure and Synthesis of Flower Pigment, Anthocyanins
Kumi Yoshida, Kin-ichi Oyama, Mihiko Mori, Tadao Kondo
Graduate School of Information Science, and Research Center for Materials Science, Nagoya
University, Chikusa, Nagoya 464-8601 Japan, and Kitasato Institute for Life Sciences, Kitasato
University, 5-9-1 Shirokane, Minato, Tokyo 108-8641, Japan.
yoshidak@is.nagoya-u.ac.jp
Enantioselective Carbon–Carbon Bond Cleavage: Rhodium-Catalyzed Restructuring
of 3-Arylcyclobutanols into 1-Indanols
Masahiro Murakami, Masanori Shigeno, Taiga Yamamoto
Department of Synthetic Chemistry and Biological Chemistry, Kyoto University, Katsura
615-8510, Japan.
murakami@sbchem.kyoto-u.ac.jp
Peptide Ligation Based on an N to S Acyl Shift Reaction
Toru Kawakami, Saburo Aimoto
Institute for Protein Research, Osaka University, 3-2 Yamadaoka, Suita, Osaka 565-0871,
Japan.
kawa@protein.osaka-u.ac.jp
Induction of Apoptosis by Rhinacanthone Isolated from Rhinacanthus nasutus Roots in
Human Cervical Carcinoma
Pongpun Siripong, Chariya Hahnvajanawong, Jantana Yahuafai, Suratsawadee Piyaviriyakul,
Kwanjai Kanokmedhakul, Ngampong Kongkathip, Somsak Ruchirawat, Naoto Oku
Natural Products Research Section, Research Division, National Cancer Institute, Bangkok
10400, Thailand; Faculty of Medicine, Khon Kaen University, Faculty of Science, Khon Kaen
University, Khon Kaen 40002, Thailand; Faculty of Science, Kasetsart University, Bangkok
10900, Thailand; Laboratory of Medicinal Chemistry, Chulabhorn Research Institute, Bangkok
10210, Thailand; and Department of Medical Biochemistry, School of Pharmaceutical Sciences,
University of Shizuoka, Shizuoka 422-8526, Japan.
pongpun8@yahoo.com
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Antimalarial and Cytotoxic Depsidones from the Fungus Chaetomium brasiliense
Somdej Kanokmedhakul, Primmala Khumkomkhet, Kwanjai Kanokmedhakul, Chariya
Hahnvajanawong, Kasem Soytong
Natural Products Research Unit, Department of Chemistry and Center for Innovation in
Chemistry, Faculty of Science, Khon Kaen University, Khon Kaen 40002, Thailand;
Department of Microbiology, and Liver Fluke and Cholangiocarcinoma Research Center,
Faculty of Medicine, Khon Kaen University, Khon Kaen 40002, Thailand; and Department of
Plant Pest Management, Faculty of Agricultural Technology, King Mongkut’s Institute of
Technology Ladkrabang, Ladkrabang, Bangkok 10520, Thailand.
somdej@kku.ac.th
Doubly Ortho-linked Quinoxaline/Spirofluorene and cis-4,4’-Bis(diarylamino)stilbene/
Fluorene Hybrids as Fluorescent Materials for Optoelectronic Applications
Chien-Tien Chen, Chin-Sheng Lin, Y. Wei, Liang-Yu Lin, Wei-San Chao
Department of Chemistry, National Taiwan Normal University, Taipei, Taiwan.
chefv043@ntnu.edu.tw
Substituted Polydonor Phthalimides: Preparation of Lariat- and Bis-Crown Ethers
Ung Chan Yoon, Dae Won Cho, Nam Kyung Sung, Hea Jung Park, Su Rhan Kim
Department of Chemistry and Chemistry Institute for Functional Materials, Pusan National
University, Busan 609-735, Korea.
ucyoon@pusan.ac.kr
Development of Activity-based Probes for Protein Tyrosine Phosphatases and Their
Applications
Yu-Yen Huang, Chun-Chen Kuo, Chi-Yuan Chu, Jing-Jer Lin, Lee-Chiang Lo
Department of Chemistry, National Taiwan University, Taipei 106, Taiwan, and Institute of
Biopharmaceutical, National Yang-Ming University, Taipei 112, Taiwan.
lclo@ntu.edu.tw
Design, Synthesis, and Biological Evaluation of 2-Phenylbenzothiazole Derivatives as
Photosensitizing Agents
Jeh-Jeng Wang, Wan-Ping Hu, Yin-Kai Chen, Chao-Cheng Liao
Department of Medicinal and Applied Chemistry, Department of Biotechnology, College of
Life Sciences, Kaohsiung Medical University, Kaohsiung, Taiwan.
jjwang@kmu.edu.tw
Evidence for a New Precursor in the Biosynthesis of the Nine-membered Enediyne Core
of the Antitumor Antibiotics C-1027
Xiaolei Chen, Zu-Feng Guo, Zhihong Guo
Department of Chemistry, Center for Cancer Research, The Hong Kong University of Science
and Technology, Clear Water Bay, Kowloon, Hong Kong SAR, China.
chguo@ust.hk
Development of the Novel Cross-linking Reaction to Thymine with High Selectivity
Fumi Nagatsugi, Tomoya Hirohama, Shuhei Kusano, Keiichi Hattori, Shuhei Imoto
Institute of Multidisciplinary Research for Advanced Materials Tohoku University, 2-1-1
Katahira, Aoba-ku, Sendai-city, Miyagi, Japan, and CREST, Japan Science and Technology
Agency.
nagatugi@tange.tohoku.ac.jp
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
8-OxoG-Clamp as a Specific Fluorescent Probe for 8-Oxoguanosine
Shigeki Sasaki, Osamu Nakagawa, Sayaka Ono, Zhichun Li, Yohei Koga
Graduate School of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi,
Higashi-ku, Fukuoka 812-8582, Japan.
sasaki@phar.kyushu-u.ac.jp
Identification of Peptide Substrate and Small Molecule Inhibitors of Testis-specific Serine/
Threonine Kinase1 (TSSK1) by the Developed Assays
Gang Liu, Leilei Zhang, Yu Yan, Zijie Liu, Abliz Zeper
Institute of Materia Medica, Chinese Academy of Medical Sciences & Peking Union Medical
College, Beijing, 100050, China.
gangliu27@yahoo.com
Insight into Inhibitor-enzyme Interactions and Structural Basis for Improving Affinity
and Potency of Novel Direct Inhibitors of the Enoyl ACP Reductase (InhA) from
Mycobacterium Tuberculosis: Molecular Modeling and Computer-aided Molecular Design
Auradee Punkvang, Patchreenart Saparpakorn, Supa Hannongbua, Peter Wolschann, Heinz
Berner, Pornpan Pungpo
Faculty of Science, Ubonratchathani University, Ubonratchathani, Thailand, 34190, Faculty
of Science, Kasetsart University, Bangkok, Thailand, 10900; Institute for Theoretical Chemistry,
University of Vienna, A-1090 Vienna, Austria; and Department of Medicinal Chemistry,
University of Vienna, A-1090 Vienna, Austria.
pornpan_ubu@yahoo.com
Synthesis and Computational Characterization of Copper Complexes of Pyridine
Derivatives with Superoxide Radical Scavenging and Antimicrobial Activities
Supaluk Prachayasittikul, Chanin Nantasenamat, Theeraphon Piacham, Chartchalerm
Isarankura-Na-Ayudhya, Virapong Prachayasitikul
Department of Clinical Microbiology, Faculty of Medical Technology, Mahidol University,
Bangkok 10700 Thailand, and Department of Chemistry, Faculty of Science, Srinakharinwirot
University, Bangkok 10110, Thailand.
mtvpr@mahidol.ac.th
Novel Anion Receptors Based on the Mixed Oligopyrrolic Macrocycles
Chang-Hee Lee
Department of Chemistry, Kangwon National University, Chun-Cheon, 200-701, Korea.
chhlee@kangwon.ac.kr
Diels-Alder Reactions of Naphthalenes in an Aqueous Molecular Host
Takashi Murase, Shinnosuke Horiuchi, Makoto Fujita
Department of Applied Chemistry, School of Engineering, The University of Tokyo, CREST,
Japan Science and Technology Agency (JST), 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-8656,
Japan.
tmurase@appchem.t.u-tokyo.ac.jp
A New Helix Electronic Theory for Molecular Chirality and Chiral Interactions and Its
Implications in Rational Design of Enantioselective Catalysis
David Zhigang Wang
School of Chemical Biology and Biotechnology, Shenzhen Graduate School of Peking
University, Shenzhen University Town, Shenzhen 518055, China.
dzw@szpku.edu.cn
The 4th International Conference on Cutting-Edge Organic Chemistry in Asia (ICCEOCA-4)
Synthesis and Theoretical Study of Molecularly Imprinted Polymers for Selective
Recognition of Antioxidants
Theeraphon Piacham, Chanin Nantasenamat, Chartchalerm Isarankura Na Ayudhya, Virapong
Prachayasittikul
Department of Clinical Microbiology, Faculty of Medical Technology, Mahidol University,
Bangkok 10700, Thailand.
mttpc@mahidol.ac.th

Source: http://www2.cri.or.th/icceoca4/ScientificProgram.pdf